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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50027046(2-[2-(3-Amino-2-hydroxy-5-methyl-hexanoylamino)-3-...)
Affinity DataKi:  900nMAssay Description:Effect of inhibitor structure on the slow binding inhibition of aminopeptidase M was determined and Ki* was reported which is obtained by the equatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50027046(2-[2-(3-Amino-2-hydroxy-5-methyl-hexanoylamino)-3-...)
Affinity DataKi:  940nMAssay Description:Compound was evaluated for the inhibitory activity against aminopeptidase MMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50027046(2-[2-(3-Amino-2-hydroxy-5-methyl-hexanoylamino)-3-...)
Affinity DataKi:  1.24E+3nMAssay Description:Compound was evaluated for the inhibition of Leucine aminopeptidase and the inhibition constant was determined after preincubating the enzyme and inh...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50027046(2-[2-(3-Amino-2-hydroxy-5-methyl-hexanoylamino)-3-...)
Affinity DataKi:  4.00E+4nMAssay Description:Effect of inhibitor structure on the slow binding inhibition of aminopeptidase M was determined and the Ki was reported which is = k2/k1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed