Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 15 hits in this display
BDBM50407517((-)ISOPROTERENOL | CHEMBL1160723 | US9492405, 27)
Ki: 46nMAssay Description:Displacement of [3H]-CGP-12177 from human beta2-adrenergic receptor expressed in CHO cells after 60 mins by radioligand competition binding assayMore data for this Ligand-Target Pair
BDBM50407517((-)ISOPROTERENOL | CHEMBL1160723 | US9492405, 27)
BDBM50407517((-)ISOPROTERENOL | CHEMBL1160723 | US9492405, 27)
BDBM50407517((-)ISOPROTERENOL | CHEMBL1160723 | US9492405, 27)
BDBM50407517((-)ISOPROTERENOL | CHEMBL1160723 | US9492405, 27)
BDBM50407517((-)ISOPROTERENOL | CHEMBL1160723 | US9492405, 27)
BDBM50407517((-)ISOPROTERENOL | CHEMBL1160723 | US9492405, 27)
BDBM50407517((-)ISOPROTERENOL | CHEMBL1160723 | US9492405, 27)
BDBM50407517((-)ISOPROTERENOL | CHEMBL1160723 | US9492405, 27)
BDBM50407517((-)ISOPROTERENOL | CHEMBL1160723 | US9492405, 27)
BDBM50407517((-)ISOPROTERENOL | CHEMBL1160723 | US9492405, 27)
BDBM50407517((-)ISOPROTERENOL | CHEMBL1160723 | US9492405, 27)
BDBM50407517((-)ISOPROTERENOL | CHEMBL1160723 | US9492405, 27)
BDBM50407517((-)ISOPROTERENOL | CHEMBL1160723 | US9492405, 27)
EC50: 2.20nMAssay Description:Activity for Beta-1 adrenergic receptor was assessed from ability to stimulate contractions in isolated guinea pig atrium.More data for this Ligand-Target Pair
BDBM50407517((-)ISOPROTERENOL | CHEMBL1160723 | US9492405, 27)