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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by
ChEMBL
Ligand
BDBM50027663
(1-(9H-Carbazol-4-yloxy)-3-isopropylamino-propan-2-...)
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Affinity Data
Ki: 0.0300nM
Assay Description:
Displacement of [3H]-CGP-12177 from human beta2-adrenergic receptor expressed in CHO cells after 60 mins by radioligand competition binding assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
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CHEMBL
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PDB
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Article
PubMed
PDB
3D Structure (crystal)
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Target
Beta-1 adrenergic receptor
(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by
ChEMBL
Ligand
BDBM50027663
(1-(9H-Carbazol-4-yloxy)-3-isopropylamino-propan-2-...)
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Affinity Data
Ki: 0.0900nM
Assay Description:
Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
PDB
Patents
Similars
In Depth
Details
Article
PubMed
PDB
3D Structure (crystal)
Copy BDB DOI
Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by
ChEMBL
Ligand
BDBM50027663
(1-(9H-Carbazol-4-yloxy)-3-isopropylamino-propan-2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.114nM
Assay Description:
Displacement of [3H]DHA from human beta2 adrenoceptor by liquid scintillation counter
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
PDB
Patents
Similars
In Depth
Details
Article
PubMed
PDB
3D Structure (crystal)
Copy BDB DOI