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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Mitogen-activated protein kinase kinase kinase 11
(Homo sapiens (Human))
Genentech
Curated by
ChEMBL
Ligand
BDBM50458548
(CHEMBL4218417)
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Affinity Data
IC50: 7nM
Assay Description:
Inhibition of recombinant GST-tagged full length human MLK3 KD expressed in baculovirus using myelin basic protein as substrate preincubated for 15 m...
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Mitogen-activated protein kinase kinase kinase 9
(Homo sapiens (Human))
Genentech
Curated by
ChEMBL
Ligand
BDBM50458548
(CHEMBL4218417)
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Copy InChI
Affinity Data
IC50: 13nM
Assay Description:
Inhibition of recombinant GST-tagged human MLK1 KD (1 to 500 residues) expressed in baculovirus using myelin basic protein as substrate preincubated ...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Mitogen-activated protein kinase kinase kinase 10
(Homo sapiens (Human))
Genentech
Curated by
ChEMBL
Ligand
BDBM50458548
(CHEMBL4218417)
Copy SMILES
Copy InChI
Affinity Data
IC50: 46nM
Assay Description:
Inhibition of recombinant GST-tagged full length human MLK2 KD/LZ expressed in baculovirus using myelin basic protein as substrate preincubated for 1...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Protein delta homolog 1
(Homo sapiens (Human))
Genentech
Curated by
ChEMBL
Ligand
BDBM50458548
(CHEMBL4218417)
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Copy InChI
Affinity Data
IC50: 119nM
Assay Description:
Inhibition of DLK (unknown origin) using myelin basic protein as substrate preincubated for 15 mins measured after 30 mins in presence of [gamma-32P]...
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI