Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chongqing Medical University

Curated by ChEMBL
LigandPNGBDBM50573595(CHEMBL4855319)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of ALK G1202R mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chongqing Medical University

Curated by ChEMBL
LigandPNGBDBM50573595(CHEMBL4855319)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chongqing Medical University

Curated by ChEMBL
LigandPNGBDBM50573595(CHEMBL4855319)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of ALK (unknown origin) preincubated for 10 mins followed by addition of substrate and ATP for 25 mins by caliper EZ reader methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Chongqing Medical University

Curated by ChEMBL
LigandPNGBDBM50573595(CHEMBL4855319)
Affinity DataIC50:  4.40nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Chongqing Medical University

Curated by ChEMBL
LigandPNGBDBM50573595(CHEMBL4855319)
Affinity DataIC50:  7.90nMAssay Description:Inhibition of recombinant human C-terminal His/FLAG-tagged HDAC1 (1 to 482 residues) expressed in Sf9 insect cells using Ac-peptide-AMC as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Chongqing Medical University

Curated by ChEMBL
LigandPNGBDBM50573595(CHEMBL4855319)
Affinity DataIC50:  9.30nMAssay Description:Inhibition of HDAC2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed