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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Mucosa-associated lymphoid tissue lymphoma translocation protein 1
(Homo sapiens (Human))
Novartis Pharma
Curated by
ChEMBL
Ligand
BDBM50555077
(CHEMBL4784806)
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Affinity Data
IC50: 15nM
Assay Description:
Inhibition of MALT1 (unknown origin) using Ac-Trp-Leu-Arg-Ser-Arg^Cys(PT14)-NH2 as substrate preincubated for 60 mins followed by substrate addition ...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Mucosa-associated lymphoid tissue lymphoma translocation protein 1
(Homo sapiens (Human))
Novartis Pharma
Curated by
ChEMBL
Ligand
BDBM50555077
(CHEMBL4784806)
Copy SMILES
Copy InChI
Affinity Data
IC50: 370nM
Assay Description:
Inhibition of MALT1 in PMA-stimulated human Jurkat T cells assessed as reduction in IL2 level pretreated for 30 mins followed by PMA-stimulation meas...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Mucosa-associated lymphoid tissue lymphoma translocation protein 1
(Homo sapiens (Human))
Novartis Pharma
Curated by
ChEMBL
Ligand
BDBM50555077
(CHEMBL4784806)
Copy SMILES
Copy InChI
Affinity Data
IC50: 5.80E+3nM
Assay Description:
Inhibition of MALT1 in human whole blood assessed as reduction in PMA//anti-CD28 antibody-induced IL2 level pre-incubated for 1 hrs before stimulatio...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI