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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284873(1-(2,6-Diisopropyl-phenyl)-3-[(4R,5R)-2-(4-hydroxy...)
Affinity DataIC50:  27nMAssay Description:Inhibitory activity against acylcoA: cholesterol acyltransferase (ACAT) in microsomes from cholesterol-fed rabbit intestinal mucosaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284873(1-(2,6-Diisopropyl-phenyl)-3-[(4R,5R)-2-(4-hydroxy...)
Affinity DataIC50:  119nMAssay Description:Inhibitory activity against acylcoA: cholesterol acyltransferase (ACAT) in microsomes from cholesterol-fed rabbit thoracic aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284873(1-(2,6-Diisopropyl-phenyl)-3-[(4R,5R)-2-(4-hydroxy...)
Affinity DataIC50:  119nMAssay Description:Inhibitory activity against acylcoA: cholesterol acyltransferase (ACAT) in microsomes from cholesterol-fed rabbit thoracic aortaMore data for this Ligand-Target Pair
In DepthDetails Article