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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50126058(2-[2-(6-Bromo-1H-indol-3-yl)-1-methyl-ethylamino]-...)
Affinity DataEC50:  38nMAssay Description:Agonism of recombinant human beta-3 adrenergic receptor assayed by measuring cAMP accumulation in CHO cells expressing beta3-ARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed