Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 7 hits in this display
BDBM258594(US9493490, 6-(4-(1-aminoethyl)-2-fluorophenoxy)ben...)
BDBM258594(US9493490, 6-(4-(1-aminoethyl)-2-fluorophenoxy)ben...)
IC50: >20nMT: 2°CAssay Description:Phosphorylation of activity of ROCK1 and ROCK2 and those of other kinases, AKT1, GRK2, PKA, PKCa and RSK1 were performed by Reaction Biology (Malvern...More data for this Ligand-Target Pair
BDBM258594(US9493490, 6-(4-(1-aminoethyl)-2-fluorophenoxy)ben...)
IC50: >30nMT: 2°CAssay Description:Phosphorylation of activity of ROCK1 and ROCK2 and those of other kinases, AKT1, GRK2, PKA, PKCa and RSK1 were performed by Reaction Biology (Malvern...More data for this Ligand-Target Pair
BDBM258594(US9493490, 6-(4-(1-aminoethyl)-2-fluorophenoxy)ben...)
IC50: >50nMT: 2°CAssay Description:Phosphorylation of activity of ROCK1 and ROCK2 and those of other kinases, AKT1, GRK2, PKA, PKCa and RSK1 were performed by Reaction Biology (Malvern...More data for this Ligand-Target Pair
BDBM258594(US9493490, 6-(4-(1-aminoethyl)-2-fluorophenoxy)ben...)
IC50: >50nMT: 2°CAssay Description:Phosphorylation of activity of ROCK1 and ROCK2 and those of other kinases, AKT1, GRK2, PKA, PKCa and RSK1 were performed by Reaction Biology (Malvern...More data for this Ligand-Target Pair
BDBM258594(US9493490, 6-(4-(1-aminoethyl)-2-fluorophenoxy)ben...)
IC50: 450nMT: 2°CAssay Description:Phosphorylation of activity of ROCK1 and ROCK2 and those of other kinases, AKT1, GRK2, PKA, PKCa and RSK1 were performed by Reaction Biology (Malvern...More data for this Ligand-Target Pair
BDBM258594(US9493490, 6-(4-(1-aminoethyl)-2-fluorophenoxy)ben...)
IC50: 540nMT: 2°CAssay Description:Phosphorylation of activity of ROCK1 and ROCK2 and those of other kinases, AKT1, GRK2, PKA, PKCa and RSK1 were performed by Reaction Biology (Malvern...More data for this Ligand-Target Pair