Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetCystine/glutamate transporter(Homo sapiens (Human))
The University Of Montana

Curated by ChEMBL

LigandBDBM50378666(CHEMBL601837)Copy SMILESCopy InChI

Affinity DataKi:  6.00E+4nMAssay Description:Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation countingMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetCystine/glutamate transporter(Homo sapiens (Human))
The University Of Montana

Curated by ChEMBL

LigandBDBM50378666(CHEMBL601837)Copy SMILESCopy InChI

Affinity DataIC50:  1.27E+5nMAssay Description:Inhibition of amino acid transport system xc- in human SNB19 cells assessed as [3H]L-glutamate uptake by liquid scintillation countingMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI