Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetCoagulation factor VII(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50148947(CHEMBL339880 | Piperidine-4-carboxylic acid [4-(1-...)
Affinity DataKi:  13nMAssay Description:In vitro inhibition of human coagulation factor VIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50148947(CHEMBL339880 | Piperidine-4-carboxylic acid [4-(1-...)
Affinity DataKi: >1.00E+4nMAssay Description:In vitro inhibition of coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50148947(CHEMBL339880 | Piperidine-4-carboxylic acid [4-(1-...)
Affinity DataKi:  6.85E+4nMAssay Description:In vitro inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed