Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetCathepsin S(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255132(4-(N-Dimethylamino)-sulfonylamino-N-[1-(2S-ethyl-4...)
Affinity DataKi:  5.30nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255132(4-(N-Dimethylamino)-sulfonylamino-N-[1-(2S-ethyl-4...)
Affinity DataKi:  300nMAssay Description:Inhibition of human recombinant cathepsin K expressed in baculovirus by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Medivir

Curated by ChEMBL
LigandPNGBDBM50255132(4-(N-Dimethylamino)-sulfonylamino-N-[1-(2S-ethyl-4...)
Affinity DataKi:  1.60E+4nMAssay Description:Inhibition of human cathepsin L by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed