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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
7
hits in this display
Target
Neuropeptide S receptor
(Homo sapiens (Human))
University Of Florida
Curated by
ChEMBL
Ligand
BDBM50511106
(CHEMBL4527708)
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Affinity Data
IC50: 3.90E+3nM
Assay Description:
Antagonist activity at human Gq-coupled NPSR1b expressed in human U2OS cells assessed as inhibition in neuropeptide S-induced beta-arrestin 2 recruit...
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Target Info
Reactome pathway
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Article
PubMed
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Target
Histamine H1 receptor
(Homo sapiens (Human))
University Of Florida
Curated by
ChEMBL
Ligand
BDBM50511106
(CHEMBL4527708)
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Affinity Data
IC50: 4.16E+3nM
Assay Description:
Antagonist activity at human Gq-coupled HRH1 expressed in CHOK1 cells assessed as inhibition in Orexin A-induced beta-arrestin 2 recruitment incubate...
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Target Info
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Article
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Target
Glucose-dependent insulinotropic receptor
(Homo sapiens (Human))
University Of Florida
Curated by
ChEMBL
Ligand
BDBM50511106
(CHEMBL4527708)
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Affinity Data
IC50: 4.62E+3nM
Assay Description:
Antagonist activity at human GPR119 expressed in human HEK293 cells assessed as inhibition in agonist-induced beta-arrestin 2 recruitment incubated f...
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Article
PubMed
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Target
Cannabinoid receptor 1
(Homo sapiens (Human))
University Of Florida
Curated by
ChEMBL
Ligand
BDBM50511106
(CHEMBL4527708)
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Affinity Data
IC50: 4.95E+3nM
Assay Description:
Antagonist activity at human Gi/o-coupled CNR1 expressed in CHOK1 cells assessed as inhibition in CP55940-induced beta-arrestin 2 recruitment incubat...
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Target Info
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Article
PubMed
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Target
Prostacyclin receptor
(Homo sapiens (Human))
University Of Florida
Curated by
ChEMBL
Ligand
BDBM50511106
(CHEMBL4527708)
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Affinity Data
IC50: 1.25E+4nM
Assay Description:
Antagonist activity at human Gs-coupled PTGIR assessed as inhibition in beraprost-induced beta-arrestin 2 recruitment incubated for 30 mins followed ...
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Target Info
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antibodypedia
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Article
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Target
Prolactin-releasing peptide receptor
(Homo sapiens (Human))
University Of Florida
Curated by
ChEMBL
Ligand
BDBM50511106
(CHEMBL4527708)
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Affinity Data
IC50: 1.38E+4nM
Assay Description:
Antagonist activity at human Gq-coupled PRLHR expressed in CHOK1 cells assessed as inhibition in prolactin releasing peptide (1 to 31)-induced beta-a...
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Target Info
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Article
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Target
Cannabinoid receptor 2
(Homo sapiens (Human))
University Of Florida
Curated by
ChEMBL
Ligand
BDBM50511106
(CHEMBL4527708)
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Affinity Data
IC50: 2.57E+4nM
Assay Description:
Antagonist activity at human Gi/o-coupled CNR2 expressed in CHOK1 cells assessed as inhibition in CP55940-induced beta-arrestin 2 recruitment incubat...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI