Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50359557(CHEMBL1927476)
Affinity DataEC50:  32nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in COS-1 cells co-transfected with Gal4 after 24 hrs by luciferase reporter gene ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50359557(CHEMBL1927476)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human PPARdelta ligand binding domain expressed in COS-1 cells after 24 hrs by luciferase reporter gene-based luminometeric analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50359557(CHEMBL1927476)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in COS-1 cells after 24 hrs by luciferase reporter gene-based luminometeric analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed