Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 100 hits in this display
IC50: 8nMAssay Description:Inhibition of human recombinant His-tagged FLT3 cytoplasmic domain (564 to 958 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 12nMAssay Description:Inhibition of human recombinant His-tagged CSF1R cytoplasmic domain (538 to 910 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 76nMAssay Description:Inhibition of human recombinant His-tagged KIT cytoplasmic domain (544 to 976 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 98nMAssay Description:Inhibition of human recombinant full length N-terminal GST/N-terminal His-tagged AMPK alpha1/beta1/gamma1 expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 157nMAssay Description:Inhibition of human recombinant His-tagged NTRK3 cytoplasmic domain (510 to 825 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 206nMAssay Description:Inhibition of human recombinant full length N-terminal GST/N-terminal His-tagged AMPK alpha2/beta1/gamma1 expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 494nMAssay Description:Inhibition of human recombinant His-tagged NTRK1 cytoplasmic domain (441 to 796 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 591nMAssay Description:Inhibition of human recombinant His-tagged FGFR2 cytoplasmic domain (403 to 822 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 668nMAssay Description:Inhibition of human recombinant full length C-terminal His-tagged SRC cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 818nMAssay Description:Inhibition of human recombinant full length C-terminal His-tagged LCK cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.01E+3nMAssay Description:Inhibition of human recombinant GST-tagged CLK2 catalytic domain (137 to 498 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.04E+3nMAssay Description:Inhibition of human recombinant GST-tagged TEK cytoplasmic domain (817 to 1101 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.15E+3nMAssay Description:Inhibition of human recombinant full length His-tagged ABL1 cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.17E+3nMAssay Description:Inhibition of human recombinant GST-tagged JAK2 cytoplasmic domain (809 to 1153 +9 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.19E+3nMAssay Description:Inhibition of human recombinant GST-tagged INSR cytoplasmic domain (1011 to 1382 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.25E+3nMAssay Description:Inhibition of human recombinant N-terminal His-tagged MET cytoplasmic domain (956 to 1390 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.26E+3nMAssay Description:Inhibition of human recombinant GST-tagged MAP3K8 catalytic domain (30 to 397 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.36E+3nMAssay Description:Inhibition of human recombinant full length His-tagged BMX cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.45E+3nMAssay Description:Inhibition of human recombinant His-tagged KDR cytoplasmic domain (789 to 1356 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.86E+3nMAssay Description:Inhibition of human full length N-terminal GST-tagged HCK cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.88E+3nMAssay Description:Inhibition of human recombinant full length His-tagged BTK cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 2.09E+3nMAssay Description:Inhibition of human recombinant His-tagged EPHA3 cytoplasmic domain (569 to 976 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 2.14E+3nMAssay Description:Inhibition of human recombinant C-terminal His-tagged IGF1R cytoplasmic domain (960 to 1397 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 2.16E+3nMAssay Description:Inhibition of human recombinant GST-tagged EPHB2 cytoplasmic domain (616 to 884 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 3.16E+3nMAssay Description:Inhibition of human recombinant GST-tagged JAK3 cytoplasmic domain (781 to 1124 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GST-tagged ALK4 catalytic domain (150 to 505 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GST-tagged PASK catalytic domain (879 to 1323 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.00E+4nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged ROCK2 cytoplasmic domain (1 to 552 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.00E+4nMAssay Description:Inhibition of human recombinant full length His-tagged ZAP70 cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.00E+4nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged TYK2 cytoplasmic domain (833 to 1187 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.00E+4nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged DAPK1 catalytic domain (1 to 363 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.00E+4nMAssay Description:Inhibition of human recombinant His-tagged ERBB2 cytoplasmic domain (676 to 1255 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GST-tagged JAK1 cytoplasmic domain (866 to 1154 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GST-tagged MINK1 catalytic domain (1 to 320 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.00E+4nMAssay Description:Inhibition of human recombinant full length His-tagged PTK6 cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GST-tagged SGK cytoplasmic domain (60 to 431 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.00E+4nMAssay Description:Inhibition of human recombinant full length N-terminal GST-tagged SYK cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GST-tagged TAOK2 cytoplasmic domain (1 to 314 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GST-tagged RPS6KB1 cytoplasmic domain (1 to 421 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GST-tagged IRAK1 catalytic domain (194 to 712 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.00E+4nMAssay Description:Inhibition of human recombinant His-tagged PRKACA catalytic domain (1 to 351 residues) expressed in Escherichia coliMore data for this Ligand-Target Pair
IC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GST-tagged EPHA8 cytoplasmic domain (565 to 1005 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.00E+4nMAssay Description:Inhibition of human recombinant full length GST-tagged ITK cytoplasmic domain expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.00E+4nMAssay Description:Inhibition of human recombinant GST-tagged ROCK1 cytoplasmic domain (1 to 535 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 1.00E+4nMAssay Description:Inhibition of human recombinant His-tagged CDC42BPA catalytic domain (1 to 473 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
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