Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 18 hits in this display
BDBM514552(US11096924, DASH-inhibitors 5349 | US11583516, Cmp...)
BDBM514552(US11096924, DASH-inhibitors 5349 | US11583516, Cmp...)
BDBM514552(US11096924, DASH-inhibitors 5349 | US11583516, Cmp...)
IC50: 250nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514552(US11096924, DASH-inhibitors 5349 | US11583516, Cmp...)
IC50: 250nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514552(US11096924, DASH-inhibitors 5349 | US11583516, Cmp...)
IC50: 610nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514552(US11096924, DASH-inhibitors 5349 | US11583516, Cmp...)
IC50: 610nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514552(US11096924, DASH-inhibitors 5349 | US11583516, Cmp...)
IC50: 730nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514552(US11096924, DASH-inhibitors 5349 | US11583516, Cmp...)
IC50: 730nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514552(US11096924, DASH-inhibitors 5349 | US11583516, Cmp...)
IC50: 3.10E+3nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514552(US11096924, DASH-inhibitors 5349 | US11583516, Cmp...)
IC50: 3.10E+3nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514552(US11096924, DASH-inhibitors 5349 | US11583516, Cmp...)
IC50: 1.40E+4nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514552(US11096924, DASH-inhibitors 5349 | US11583516, Cmp...)
IC50: 1.40E+4nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514552(US11096924, DASH-inhibitors 5349 | US11583516, Cmp...)
BDBM514552(US11096924, DASH-inhibitors 5349 | US11583516, Cmp...)
IC50: 2.50E+5nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM514552(US11096924, DASH-inhibitors 5349 | US11583516, Cmp...)
IC50: 6.10E+5nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM514552(US11096924, DASH-inhibitors 5349 | US11583516, Cmp...)
IC50: 7.30E+5nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM514552(US11096924, DASH-inhibitors 5349 | US11583516, Cmp...)
IC50: 3.10E+6nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM514552(US11096924, DASH-inhibitors 5349 | US11583516, Cmp...)
IC50: 1.40E+7nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair