Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 21 hits in this display
BDBM514554(US11096924, DASH-inhibitors 5363 | US11583516, Cmp...)
BDBM514554(US11096924, DASH-inhibitors 5363 | US11583516, Cmp...)
BDBM514554(US11096924, DASH-inhibitors 5363 | US11583516, Cmp...)
IC50: 5.20nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514554(US11096924, DASH-inhibitors 5363 | US11583516, Cmp...)
IC50: 5.20nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514554(US11096924, DASH-inhibitors 5363 | US11583516, Cmp...)
IC50: 5.5nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514554(US11096924, DASH-inhibitors 5363 | US11583516, Cmp...)
IC50: 5.5nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514554(US11096924, DASH-inhibitors 5363 | US11583516, Cmp...)
IC50: 32nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514554(US11096924, DASH-inhibitors 5363 | US11583516, Cmp...)
IC50: 32nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514554(US11096924, DASH-inhibitors 5363 | US11583516, Cmp...)
IC50: 110nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514554(US11096924, DASH-inhibitors 5363 | US11583516, Cmp...)
IC50: 110nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514554(US11096924, DASH-inhibitors 5363 | US11583516, Cmp...)
IC50: 270nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514554(US11096924, DASH-inhibitors 5363 | US11583516, Cmp...)
IC50: 270nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514554(US11096924, DASH-inhibitors 5363 | US11583516, Cmp...)
IC50: 1.40E+3nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514554(US11096924, DASH-inhibitors 5363 | US11583516, Cmp...)
BDBM514554(US11096924, DASH-inhibitors 5363 | US11583516, Cmp...)
IC50: 1.40E+3nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514554(US11096924, DASH-inhibitors 5363 | US11583516, Cmp...)
IC50: 5.20E+3nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM514554(US11096924, DASH-inhibitors 5363 | US11583516, Cmp...)
IC50: 5.50E+3nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM514554(US11096924, DASH-inhibitors 5363 | US11583516, Cmp...)
IC50: 3.20E+4nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM514554(US11096924, DASH-inhibitors 5363 | US11583516, Cmp...)
IC50: 1.10E+5nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM514554(US11096924, DASH-inhibitors 5363 | US11583516, Cmp...)
IC50: 2.70E+5nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM514554(US11096924, DASH-inhibitors 5363 | US11583516, Cmp...)
IC50: 1.40E+6nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair