Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 6 hits in this display
BDBM50045598(CHEMBL3314311 | US9540323, 220 | US9540323, exampl...)
BDBM50045598(CHEMBL3314311 | US9540323, 220 | US9540323, exampl...)
Ki: 14nM ΔG°: -44.8kJ/molepH: 7.4 T: 2°CAssay Description:A SPA membrane binding assay was used to identify inhibitors of [33P] 2MeS-ADP binding to cloned human P2Y1 receptors (The P2Y1 receptor membranes we...More data for this Ligand-Target Pair
BDBM50045598(CHEMBL3314311 | US9540323, 220 | US9540323, exampl...)
BDBM50045598(CHEMBL3314311 | US9540323, 220 | US9540323, exampl...)
IC50: 1.10nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
BDBM50045598(CHEMBL3314311 | US9540323, 220 | US9540323, exampl...)
BDBM50045598(CHEMBL3314311 | US9540323, 220 | US9540323, exampl...)