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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

TargetCarbonic anhydrase 2(Homo sapiens (Human))
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50208749(1-[2-(4-sulfamoylphenyl)ethyl]-3-{[(1R,2S,6S,9R)-4...)
Affinity DataKi:  10nMAssay Description:Inhibition of human recombinant CA2 after 15 mins by CO2 hydration stopped flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50208749(1-[2-(4-sulfamoylphenyl)ethyl]-3-{[(1R,2S,6S,9R)-4...)
Affinity DataKi:  10nMAssay Description:Inhibition of human recombinant CA9 after 15 mins by CO2 hydration stopped flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50208749(1-[2-(4-sulfamoylphenyl)ethyl]-3-{[(1R,2S,6S,9R)-4...)
Affinity DataKi:  24nMAssay Description:Inhibition of human recombinant CA7 after 15 mins by CO2 hydration stopped flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 4(Homo sapiens (Human))
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50208749(1-[2-(4-sulfamoylphenyl)ethyl]-3-{[(1R,2S,6S,9R)-4...)
Affinity DataKi:  850nMAssay Description:Inhibition of human recombinant CA4 after 15 mins by CO2 hydration stopped flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 14(Homo sapiens (Human))
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50208749(1-[2-(4-sulfamoylphenyl)ethyl]-3-{[(1R,2S,6S,9R)-4...)
Affinity DataKi:  2.35E+3nMAssay Description:Inhibition of human recombinant CA14 after 15 mins by CO2 hydration stopped flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50208749(1-[2-(4-sulfamoylphenyl)ethyl]-3-{[(1R,2S,6S,9R)-4...)
Affinity DataKi:  1.07E+4nMAssay Description:Inhibition of human recombinant CA1 after 15 mins by CO2 hydration stopped flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50208749(1-[2-(4-sulfamoylphenyl)ethyl]-3-{[(1R,2S,6S,9R)-4...)
Affinity DataKi:  3.98E+4nMAssay Description:Inhibition of human recombinant CA5A after 15 mins by CO2 hydration stopped flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed