Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 300 hits in this display
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 3.80nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 3.80nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 incubated for 15 mins prior to testing by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 6.60nMAssay Description:Inhibition of recombinant Sulfurihydrogenibium yellowstonense YO3AOP1 carbonic anhydrase by stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 10nMAssay Description:Inhibition of human recombinant cytosolic carbonic anhydrase 2 pre-incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 10nMAssay Description:Inhibition of recombinant human carbonic anhydrase 2 incubated for 15 mins prior to testing by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 10nMAssay Description:Inhibition of human recombinant Carbonic anhydrase 2 compound preincubated for 15 mins by stopped flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 10nMAssay Description:Inhibition of human Carbonic anhydrase2 using CO2 as substrate preincubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 10nMAssay Description:Inhibition of human wild type carbonic anhydrase 2 expressed in Escherichia coli after 15 mins preincubation by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 30nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 30nM ΔG°: -42.9kJ/molepH: 7.4 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 45nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 47nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 58nMAssay Description:Inhibition of human recombinant CA9 catalytic domain-mediated CO2 hydration preincubated for 15 mins by stopped-flow assayMore data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 58nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 58nM ΔG°: -40.9kJ/molepH: 7.5 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 58nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 63nM ΔG°: -41.1kJ/molepH: 7.4 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 78nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 250nM ΔG°: -37.3kJ/molepH: 7.5 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 250nM ΔG°: -37.7kJ/molepH: 7.4 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 250nMAssay Description:Inhibition of human recombinant Carbonic anhydrase 1 compound preincubated for 15 mins by stopped flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 250nMAssay Description:Inhibition of human Carbonic anhydrase1 using CO2 as substrate preincubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 250nMAssay Description:Inhibition of wild type human recombinant carbonic anhydrase 1 expressed in Escherichia coli BL21 (DE3) after 15 mins by CO2 hydration methodMore data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 250nMAssay Description:Inhibition of human recombinant cytosolic carbonic anhydrase 1 pre-incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 250nMAssay Description:Inhibition of recombinant human carbonic anhydrase 1 incubated for 15 mins prior to testing by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Carbonic anhydrase(Cryptococcus neoformans var. grubii (Filobasidiell...)Universite Degli Studi Di Firenze
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Carbonic anhydrase(Cryptococcus neoformans var. grubii (Filobasidiell...)Universite Degli Studi Di Firenze
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 370nMAssay Description:Inhibition of Cryptococcus neoformans recombinant Can2 beta-carbonic anhydrase after 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 392nMAssay Description:Inhibition of Thalassiosira weissflogii delta carbonic anhydrase preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 474nMAssay Description:Inhibition of full length Mycobacterium tuberculosis H37Rv recombinant carbonic anhydrase 2 encoded by RV3588c by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 610nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant Rv1284 beta-carbonic anhydrase after 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 1.11E+3nMAssay Description:Inhibition of Candida albicans recombinant Nce103 beta-carbonic anhydrase after 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 1.46E+3nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 1.46E+3nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 1.46E+3nMAssay Description:Inhibition of human recombinant full length CA14-mediated CO2 hydration preincubated for 15 mins by stopped-flow assayMore data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 3.02E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant Rv3273 beta-carbonic anhydrase after 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 4.90E+3nMAssay Description:Inhibition of truncated human cloned membrane-associated carbonic anhydrase 4 preincubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 4.90E+3nM ΔG°: -30.3kJ/molepH: 7.4 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 4.90E+3nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 3.00E+4nMAssay Description:Inhibition of full length human recombinant mitochondrial carbonic anhydrase 5B preincubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 6.30E+4nMAssay Description:Inhibition of full length human recombinant mitochondrial carbonic anhydrase 5A pre-incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Ki: 7.80E+5nM ΔG°: -17.7kJ/molepH: 7.4 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Kd: 290nMpH: 7.5Assay Description:Binding affinity to human carbonic anhydrase 2 in presence of 10 mM HEPES and 100 uM Na2SO4 at pH 7.5 by ThermoFluor methodMore data for this Ligand-Target Pair
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
BDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
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