Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 21 hits in this display
BDBM514520(US11096924, DASH-inhibitors 4175 CP | US11583516, ...)
BDBM514520(US11096924, DASH-inhibitors 4175 CP | US11583516, ...)
BDBM514520(US11096924, DASH-inhibitors 4175 CP | US11583516, ...)
IC50: 5.30nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514520(US11096924, DASH-inhibitors 4175 CP | US11583516, ...)
IC50: 5.30nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514520(US11096924, DASH-inhibitors 4175 CP | US11583516, ...)
IC50: 5.60nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514520(US11096924, DASH-inhibitors 4175 CP | US11583516, ...)
IC50: 5.60nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514520(US11096924, DASH-inhibitors 4175 CP | US11583516, ...)
IC50: 9.20nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514520(US11096924, DASH-inhibitors 4175 CP | US11583516, ...)
IC50: 9.20nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514520(US11096924, DASH-inhibitors 4175 CP | US11583516, ...)
IC50: 27nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514520(US11096924, DASH-inhibitors 4175 CP | US11583516, ...)
IC50: 27nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514520(US11096924, DASH-inhibitors 4175 CP | US11583516, ...)
IC50: 68nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514520(US11096924, DASH-inhibitors 4175 CP | US11583516, ...)
IC50: 68nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514520(US11096924, DASH-inhibitors 4175 CP | US11583516, ...)
IC50: 88nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514520(US11096924, DASH-inhibitors 4175 CP | US11583516, ...)
IC50: 88nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514520(US11096924, DASH-inhibitors 4175 CP | US11583516, ...)
BDBM514520(US11096924, DASH-inhibitors 4175 CP | US11583516, ...)
IC50: 5.30E+3nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM514520(US11096924, DASH-inhibitors 4175 CP | US11583516, ...)
IC50: 5.60E+3nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM514520(US11096924, DASH-inhibitors 4175 CP | US11583516, ...)
IC50: 9.20E+3nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM514520(US11096924, DASH-inhibitors 4175 CP | US11583516, ...)
IC50: 2.70E+4nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM514520(US11096924, DASH-inhibitors 4175 CP | US11583516, ...)
IC50: 6.80E+4nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM514520(US11096924, DASH-inhibitors 4175 CP | US11583516, ...)
IC50: 8.80E+4nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair