Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 21 hits in this display
BDBM514516(US11096924, DASH-inhibitors 4175 CH | US11583516, ...)
BDBM514516(US11096924, DASH-inhibitors 4175 CH | US11583516, ...)
BDBM514516(US11096924, DASH-inhibitors 4175 CH | US11583516, ...)
IC50: 2.80nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514516(US11096924, DASH-inhibitors 4175 CH | US11583516, ...)
IC50: 2.80nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514516(US11096924, DASH-inhibitors 4175 CH | US11583516, ...)
IC50: 5.40nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514516(US11096924, DASH-inhibitors 4175 CH | US11583516, ...)
IC50: 5.40nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514516(US11096924, DASH-inhibitors 4175 CH | US11583516, ...)
IC50: 5.80nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514516(US11096924, DASH-inhibitors 4175 CH | US11583516, ...)
IC50: 5.80nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514516(US11096924, DASH-inhibitors 4175 CH | US11583516, ...)
IC50: 34nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514516(US11096924, DASH-inhibitors 4175 CH | US11583516, ...)
IC50: 34nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514516(US11096924, DASH-inhibitors 4175 CH | US11583516, ...)
IC50: 54nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514516(US11096924, DASH-inhibitors 4175 CH | US11583516, ...)
IC50: 54nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514516(US11096924, DASH-inhibitors 4175 CH | US11583516, ...)
IC50: 76nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM514516(US11096924, DASH-inhibitors 4175 CH | US11583516, ...)
IC50: 76nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
BDBM514516(US11096924, DASH-inhibitors 4175 CH | US11583516, ...)
BDBM514516(US11096924, DASH-inhibitors 4175 CH | US11583516, ...)
IC50: 2.80E+3nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM514516(US11096924, DASH-inhibitors 4175 CH | US11583516, ...)
IC50: 5.40E+3nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM514516(US11096924, DASH-inhibitors 4175 CH | US11583516, ...)
IC50: 5.80E+3nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM514516(US11096924, DASH-inhibitors 4175 CH | US11583516, ...)
IC50: 3.40E+4nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM514516(US11096924, DASH-inhibitors 4175 CH | US11583516, ...)
IC50: 5.40E+4nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM514516(US11096924, DASH-inhibitors 4175 CH | US11583516, ...)
IC50: 7.60E+4nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair