Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 14 hits in this display
BDBM50173320(GSK-180736A | GSK180736A | US10023564, Compound GS...)
BDBM50173320(GSK-180736A | GSK180736A | US10023564, Compound GS...)
BDBM50173320(GSK-180736A | GSK180736A | US10023564, Compound GS...)
BDBM50173320(GSK-180736A | GSK180736A | US10023564, Compound GS...)
BDBM50173320(GSK-180736A | GSK180736A | US10023564, Compound GS...)
BDBM50173320(GSK-180736A | GSK180736A | US10023564, Compound GS...)
BDBM50173320(GSK-180736A | GSK180736A | US10023564, Compound GS...)
BDBM50173320(GSK-180736A | GSK180736A | US10023564, Compound GS...)
IC50: 1.00E+5nMpH: 7.0Assay Description:GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e...More data for this Ligand-Target Pair
BDBM50173320(GSK-180736A | GSK180736A | US10023564, Compound GS...)
BDBM50173320(GSK-180736A | GSK180736A | US10023564, Compound GS...)
BDBM50173320(GSK-180736A | GSK180736A | US10023564, Compound GS...)
IC50: >1.00E+5nMpH: 7.0Assay Description:GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e...More data for this Ligand-Target Pair
BDBM50173320(GSK-180736A | GSK180736A | US10023564, Compound GS...)
BDBM50173320(GSK-180736A | GSK180736A | US10023564, Compound GS...)
BDBM50173320(GSK-180736A | GSK180736A | US10023564, Compound GS...)
IC50: >1.00E+6nMAssay Description:Inhibition of bovine GRK1 (1 to 535 residues) assessed as decrease in phosphorylation of tubulin after 5 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair