Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetCoagulation factor X(Homo sapiens (Human))
Southern Research

Curated by ChEMBL
LigandPNGBDBM50157632(CHEMBL3781349)
Affinity DataKi:  380nMAssay Description:Inhibition of human recombinant factor 10a using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Southern Research

Curated by ChEMBL
LigandPNGBDBM50157632(CHEMBL3781349)
Affinity DataKi:  430nMAssay Description:Inhibition of human recombinant trypsin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor activator(Homo sapiens (Human))
Southern Research

Curated by ChEMBL
LigandPNGBDBM50157632(CHEMBL3781349)
Affinity DataKi:  480nMAssay Description:Inhibition of human recombinant hepatocyte growth factor activator using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Southern Research

Curated by ChEMBL
LigandPNGBDBM50157632(CHEMBL3781349)
Affinity DataKi:  530nMAssay Description:Inhibition of human recombinant matripase catalytic domain using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease hepsin(Homo sapiens (Human))
Southern Research

Curated by ChEMBL
LigandPNGBDBM50157632(CHEMBL3781349)
Affinity DataKi:  540nMAssay Description:Inhibition of human recombinant hepsin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Southern Research

Curated by ChEMBL
LigandPNGBDBM50157632(CHEMBL3781349)
Affinity DataKi:  1.16E+4nMAssay Description:Inhibition of human recombinant thrombin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed