Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetPepsin A(Porcine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50141614((1S,2S,5S)-3-Hydroxy-4-[2-((S)-hydroxy-6-(S)-4-{(S...)
Affinity DataKi:  0.0460nMAssay Description:Inhibitory activity of the compound against aspartyl protease pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPepsin A(Porcine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50022866(4-[1-{3-[1-[1-(1-amino-1-methylpropylcarboxamido)-...)
Affinity DataIC50:  11nMAssay Description:Inhibitory activity against porcine pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Bos taurus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50022866(4-[1-{3-[1-[1-(1-amino-1-methylpropylcarboxamido)-...)
Affinity DataIC50:  46nMAssay Description:Inhibitory activity against bovine cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin-1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50022866(4-[1-{3-[1-[1-(1-amino-1-methylpropylcarboxamido)-...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibitory activity against mouse reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50022866(4-[1-{3-[1-[1-(1-amino-1-methylpropylcarboxamido)-...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibitory activity against human reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed