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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetEnteropeptidase(Homo sapiens (Human))
Ajinomoto

US Patent
LigandPNGBDBM158138(US9024044, 66 | US9227949, 66 | US9655879, 66)
Affinity DataKi:  0.710nMpH: 8.0Assay Description:Using a 96 well plate (#3915, Costar), a test compound (25 uL), 400 mM Tris-HCl buffer (pH 8.0, 25 uL) and 0.5 mg/mL, fluorescence enzyme substrate (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEnteropeptidase(Homo sapiens (Human))
Ajinomoto

US Patent
LigandPNGBDBM158138(US9024044, 66 | US9227949, 66 | US9655879, 66)
Affinity DataKi:  0.710nMAssay Description:Using a 96 well plate (#3915, Costar), a test compound (25 μL) was mixed with 20 μM fluorescence enzyme substrate (Boc-Phe-Ser-Arg-AMC, 50 ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEnteropeptidase(Homo sapiens (Human))
Ajinomoto

US Patent
LigandPNGBDBM158138(US9024044, 66 | US9227949, 66 | US9655879, 66)
Affinity DataKi:  0.710nMpH: 8.0Assay Description:Using a 96 well plate (#3915, Costar), a test compound (25 μL), 400 mM Tris-HCl buffer (pH 8.0, 25 μL) and 0.5 mg/mL fluorescence enzyme su...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Ea Pharma

US Patent
LigandPNGBDBM158138(US9024044, 66 | US9227949, 66 | US9655879, 66)
Affinity DataKi:  1.58nMAssay Description:Using a 96 well plate (#3915, Costar), a test compound (25 μL), 400 mM Tris-HCl buffer (pH 8.0, 25 μL) and 0.5 mg/mL fluorescence enzyme su...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Ea Pharma

US Patent
LigandPNGBDBM158138(US9024044, 66 | US9227949, 66 | US9655879, 66)
Affinity DataKi:  1.58nMpH: 8.0Assay Description:Using a 96 well plate (#3915, Costar), a test compound (25 uL) was mixed with 20 uM fluorescence enzyme substrate (Boc-Phe-Ser-Arg-AMC, 50 uL) mixed ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Ea Pharma

US Patent
LigandPNGBDBM158138(US9024044, 66 | US9227949, 66 | US9655879, 66)
Affinity DataKi:  1.58nMpH: 8.0Assay Description:Using a 96 well plate (#3915, Costar), a test compound (25 μL) was mixed with 20 μM fluorescence enzyme substrate (Boc-Phe-Ser-Arg-AMC, 50 ...More data for this Ligand-Target Pair
In DepthDetails US Patent