Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 14 hits in this display
BDBM50017716(2,2-Diphenyl-pentanoic acid 2-diethylamino-ethyl e...)
BDBM50017716(2,2-Diphenyl-pentanoic acid 2-diethylamino-ethyl e...)
BDBM50017716(2,2-Diphenyl-pentanoic acid 2-diethylamino-ethyl e...)
BDBM50017716(2,2-Diphenyl-pentanoic acid 2-diethylamino-ethyl e...)
BDBM50017716(2,2-Diphenyl-pentanoic acid 2-diethylamino-ethyl e...)
BDBM50017716(2,2-Diphenyl-pentanoic acid 2-diethylamino-ethyl e...)
BDBM50017716(2,2-Diphenyl-pentanoic acid 2-diethylamino-ethyl e...)
BDBM50017716(2,2-Diphenyl-pentanoic acid 2-diethylamino-ethyl e...)
BDBM50017716(2,2-Diphenyl-pentanoic acid 2-diethylamino-ethyl e...)
BDBM50017716(2,2-Diphenyl-pentanoic acid 2-diethylamino-ethyl e...)
BDBM50017716(2,2-Diphenyl-pentanoic acid 2-diethylamino-ethyl e...)
EC50: 1.26E+4nMAssay Description:Activation of human PXR expressed in human HepG2 (DPX-2) cells assessed as induction of CYP3A4 after 24 hrs by luminescent analysisMore data for this Ligand-Target Pair
BDBM50017716(2,2-Diphenyl-pentanoic acid 2-diethylamino-ethyl e...)
BDBM50017716(2,2-Diphenyl-pentanoic acid 2-diethylamino-ethyl e...)
EC50: 3.55E+4nMAssay Description:Activation of rat PXR expressed in human HepG2 cells after 24 hrs by luciferase reporter gene based luminescent analysisMore data for this Ligand-Target Pair
BDBM50017716(2,2-Diphenyl-pentanoic acid 2-diethylamino-ethyl e...)
EC50: 2.51E+4nMAssay Description:Activation of human PXR expressed in human HepG2 (DPX-2) cells after 24 hrs by luciferase reporter gene based luminescent analysisMore data for this Ligand-Target Pair