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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Histamine H3 receptor
(Homo sapiens (Human))
Jagiellonian University Medical College
Curated by
ChEMBL
Ligand
BDBM50074088
((2-Methyl-pentyl)-carbamic acid 3-(1H-imidazol-4-y...)
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Affinity Data
Ki: 8.30nM
Assay Description:
Displacement of [3H]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Histamine H3 receptor
(Rattus norvegicus (rat))
Freie UniversitäT Berlin
Curated by
ChEMBL
Ligand
BDBM50074088
((2-Methyl-pentyl)-carbamic acid 3-(1H-imidazol-4-y...)
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Affinity Data
Ki: 15nM
Assay Description:
Effect at histamine H3 receptors (in vitro) on synaptosomes of rat cerebral cortex assayed by functional H3-receptor assay.
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Histamine H3 receptor
(Rattus norvegicus (rat))
Freie UniversitäT Berlin
Curated by
ChEMBL
Ligand
BDBM50074088
((2-Methyl-pentyl)-carbamic acid 3-(1H-imidazol-4-y...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 15nM
Assay Description:
Displacement of [3H]histamine from histamine H3 receptor in rat cerebral cortex
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Histamine H4 receptor
(Homo sapiens (Human))
Jagiellonian University Medical College
Curated by
ChEMBL
Ligand
BDBM50074088
((2-Methyl-pentyl)-carbamic acid 3-(1H-imidazol-4-y...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 162nM
Assay Description:
Displacement of [3H]histamine from human histamine H4 receptor expressed in SF9 cells coexpressing Galphai2, Gbeta1gamma2
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI