Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 7 hits in this display
Cathepsin S(Homo sapiens (Human))University of California Berkeley
BDBM19483(1, 2, 3 -Triazole Nitrile Inhibitor, 11d | N-[(1S)...)
Cathepsin K(Homo sapiens (Human))University of California Berkeley
BDBM19483(1, 2, 3 -Triazole Nitrile Inhibitor, 11d | N-[(1S)...)
Ki: 1.70E+3nM ΔG°: -34.3kJ/molepH: 6.1 T: 2°CAssay Description:The proteolytic cleavage of N-acyl aminocoumarins by cathepsins was conducted in Dynatech Microfluor fluorescence 96-well microtiter plates, and read...More data for this Ligand-Target Pair
BDBM19483(1, 2, 3 -Triazole Nitrile Inhibitor, 11d | N-[(1S)...)
Ki: >1.00E+4nM ΔG°: >-29.7kJ/molepH: 6.1 T: 2°CAssay Description:The proteolytic cleavage of N-acyl aminocoumarins by cathepsins was conducted in Dynatech Microfluor fluorescence 96-well microtiter plates, and read...More data for this Ligand-Target Pair
Cathepsin B(Homo sapiens (Human))University of California Berkeley
BDBM19483(1, 2, 3 -Triazole Nitrile Inhibitor, 11d | N-[(1S)...)
Ki: >1.00E+4nM ΔG°: >-29.7kJ/molepH: 6.1 T: 2°CAssay Description:The proteolytic cleavage of N-acyl aminocoumarins by cathepsins was conducted in Dynatech Microfluor fluorescence 96-well microtiter plates, and read...More data for this Ligand-Target Pair
Cathepsin S(Homo sapiens (Human))University of California Berkeley
BDBM19483(1, 2, 3 -Triazole Nitrile Inhibitor, 11d | N-[(1S)...)
Cathepsin S(Homo sapiens (Human))University of California Berkeley
BDBM19483(1, 2, 3 -Triazole Nitrile Inhibitor, 11d | N-[(1S)...)
BDBM19483(1, 2, 3 -Triazole Nitrile Inhibitor, 11d | N-[(1S)...)