Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetPancreatic alpha-amylase(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033631(2-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  0.300nMAssay Description:Tested in vitro for inhibition of amylase release from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033631(2-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  7nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033631(2-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  210nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033631(2-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  500nMAssay Description:Tested in vitro for amylase release from rat pancreatic acini (percent of secretion)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed