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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetGastrin/cholecystokinin type B receptor(RAT)
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033633(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  12nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033633(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  15nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033633(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  32nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033633(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  75nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033633(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  190nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033633(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  205nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033633(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataEC50:  6nMAssay Description:Tested for inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033633(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataEC50:  50nMAssay Description:Tested in vitro for amylase release from rat pancreatic acini (percent of secretion)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed