Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetHistone deacetylase 6(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50268605(CHEMBL4086409)
Affinity DataIC50:  320nMAssay Description:Inhibition of HDAC6 (unknown origin) by ELISA-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50268605(CHEMBL4086409)
Affinity DataIC50:  430nMAssay Description:Inhibition of HDAC8 (unknown origin) by ELISA-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50268605(CHEMBL4086409)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of HDAC1 (unknown origin) by ELISA-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50268605(CHEMBL4086409)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of HDAC2 (unknown origin) by ELISA-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50268605(CHEMBL4086409)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of HDAC3 (unknown origin) by ELISA-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed