Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 12 hits in this display
BDBM50191588((2R,3S,6S,7R,8R)-3-[(3-formamido-2-hydroxybenzoyl)...)
BDBM50191588((2R,3S,6S,7R,8R)-3-[(3-formamido-2-hydroxybenzoyl)...)
BDBM50191588((2R,3S,6S,7R,8R)-3-[(3-formamido-2-hydroxybenzoyl)...)
IC50: 2nMAssay Description:Inhibition of Septoria nodorum succinate dehydrogenase and Qi site of mitochondrial respiratory chain complex 3 by FMET2-3 assayMore data for this Ligand-Target Pair
Cytochrome b(Candida albicans (Yeast))Massachusetts Institute of Technology
BDBM192008(Antimycin A | [(2R,3S,6S,7R)-3-[(3-formamido-2-hyd...)
Cytochrome b(Homo sapiens (Human))Massachusetts Institute of Technology
BDBM192008(Antimycin A | [(2R,3S,6S,7R)-3-[(3-formamido-2-hyd...)
IC50: 7nMpH: 7.4 T: 2°CAssay Description:The cytochrome b enzyme assay was adapted from previous studies (Gutierrez-Cirlos et al., 2004). Briefly, compounds were diluted in a 23 reaction buf...More data for this Ligand-Target Pair
BDBM50191588((2R,3S,6S,7R,8R)-3-[(3-formamido-2-hydroxybenzoyl)...)
BDBM50191588((2R,3S,6S,7R,8R)-3-[(3-formamido-2-hydroxybenzoyl)...)
BDBM50191588((2R,3S,6S,7R,8R)-3-[(3-formamido-2-hydroxybenzoyl)...)
BDBM50191588((2R,3S,6S,7R,8R)-3-[(3-formamido-2-hydroxybenzoyl)...)
BDBM50191588((2R,3S,6S,7R,8R)-3-[(3-formamido-2-hydroxybenzoyl)...)
BDBM50191588((2R,3S,6S,7R,8R)-3-[(3-formamido-2-hydroxybenzoyl)...)
BDBM50191588((2R,3S,6S,7R,8R)-3-[(3-formamido-2-hydroxybenzoyl)...)