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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetProlyl endopeptidase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50240495((R)-1-(4-(pyrrolidine-1-carbonyl)thiazolidin-3-yl)...)
Affinity DataIC50:  11nMAssay Description:Inhibitory activity against rat brain Prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50240495((R)-1-(4-(pyrrolidine-1-carbonyl)thiazolidin-3-yl)...)
Affinity DataIC50:  11nMAssay Description:Inhibition of POP in Sprague-Dawley rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed