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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
26
hits in this display
Target
Probable G-protein coupled receptor 34
(Homo sapiens (Human))
The University Of Tokyo
Curated by
ChEMBL
Ligand
BDBM50096349
(CHEBI:52649 | CHEMBL1742484)
Copy SMILES
Copy InChI
Affinity Data
EC50: 550nM
Assay Description:
Agonist activity at GPR34 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Probable G-protein coupled receptor 174
(Mus musculus)
The University Of Tokyo
Curated by
ChEMBL
Ligand
BDBM50096349
(CHEBI:52649 | CHEMBL1742484)
Copy SMILES
Copy InChI
Affinity Data
EC50: 34nM
Assay Description:
Agonist activity at mouse GPR174 transfected in human HEK293FT cells co-transfected with AP-TGFalpha assessed as AP-TGFalpha release incubated for 90...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
PubMed
Copy BDB DOI
Target
Probable G-protein coupled receptor 174
(Homo sapiens (Human))
The University Of Tokyo
Curated by
ChEMBL
Ligand
BDBM50096349
(CHEBI:52649 | CHEMBL1742484)
Copy SMILES
Copy InChI
Affinity Data
EC50: 525nM
Assay Description:
Agonist activity at GPR174 (unknown origin) transfected in HEK293FT cells after 1 hr by TGFalpha shedding assay
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Probable G-protein coupled receptor 34
(Homo sapiens (Human))
The University Of Tokyo
Curated by
ChEMBL
Ligand
BDBM50096349
(CHEBI:52649 | CHEMBL1742484)
Copy SMILES
Copy InChI
Affinity Data
EC50: 550nM
Assay Description:
Agonist activity at GPR34 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Putative P2Y purinoceptor 10
(Homo sapiens (Human))
The University Of Tokyo
Curated by
ChEMBL
Ligand
BDBM50096349
(CHEBI:52649 | CHEMBL1742484)
Copy SMILES
Copy InChI
Affinity Data
EC50: 28nM
Assay Description:
Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay
More data for this Ligand-Target Pair
Target Info
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Probable G-protein coupled receptor 174
(Homo sapiens (Human))
The University Of Tokyo
Curated by
ChEMBL
Ligand
BDBM50096349
(CHEBI:52649 | CHEMBL1742484)
Copy SMILES
Copy InChI
Affinity Data
EC50: 520nM
Assay Description:
Agonist activity at GPR174 (unknown origin) transfected in HEK293FT cells after 1 hr by TGFalpha shedding assay
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Probable G-protein coupled receptor 34
(Mus musculus)
The University Of Tokyo
Curated by
ChEMBL
Ligand
BDBM50096349
(CHEBI:52649 | CHEMBL1742484)
Copy SMILES
Copy InChI
Affinity Data
EC50: 240nM
Assay Description:
Agonist activity at mouse GPR34 expressed in HEK293A cells cotransfected with chimeric Galphaq/il after 1.5 hrs by alkaline phosphatase tagged-TGFalp...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Putative P2Y purinoceptor 10
(Mus musculus)
The University Of Tokyo
Curated by
ChEMBL
Ligand
BDBM50096349
(CHEBI:52649 | CHEMBL1742484)
Copy SMILES
Copy InChI
Affinity Data
EC50: 25nM
Assay Description:
Agonist activity at mouse P2Y10 receptor expressed in HEK293A cells after 1.5 hrs by alkaline phosphatase tagged-TGFalpha shedding assay
More data for this Ligand-Target Pair
Target Info
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Putative P2Y purinoceptor 10
(Mus musculus)
The University Of Tokyo
Curated by
ChEMBL
Ligand
BDBM50096349
(CHEBI:52649 | CHEMBL1742484)
Copy SMILES
Copy InChI
Affinity Data
EC50: 25nM
Assay Description:
Agonist activity at mouse P2Y10 receptor expressed in HEK293A cells after 1.5 hrs by alkaline phosphatase tagged-TGFalpha shedding assay
More data for this Ligand-Target Pair
Target Info
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Probable G-protein coupled receptor 34
(Mus musculus)
The University Of Tokyo
Curated by
ChEMBL
Ligand
BDBM50096349
(CHEBI:52649 | CHEMBL1742484)
Copy SMILES
Copy InChI
Affinity Data
EC50: 240nM
Assay Description:
Agonist activity at mouse GPR34 expressed in HEK293A cells cotransfected with chimeric Galphaq/il after 1.5 hrs by alkaline phosphatase tagged-TGFalp...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Probable G-protein coupled receptor 34
(Mus musculus)
The University Of Tokyo
Curated by
ChEMBL
Ligand
BDBM50096349
(CHEBI:52649 | CHEMBL1742484)
Copy SMILES
Copy InChI
Affinity Data
EC50: 417nM
Assay Description:
Agonist activity at mouse GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/chimeric Galphaq/i1 assessed as induction of ectodomain she...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Probable G-protein coupled receptor 34
(Homo sapiens (Human))
The University Of Tokyo
Curated by
ChEMBL
Ligand
BDBM50096349
(CHEBI:52649 | CHEMBL1742484)
Copy SMILES
Copy InChI
Affinity Data
EC50: 250nM
Assay Description:
Agonist activity at human GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/chimeric Galphaq/i1 assessed as induction of AP-TGFalpha re...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Probable G-protein coupled receptor 34
(Mus musculus)
The University Of Tokyo
Curated by
ChEMBL
Ligand
BDBM50096349
(CHEBI:52649 | CHEMBL1742484)
Copy SMILES
Copy InChI
Affinity Data
EC50: 420nM
Assay Description:
Agonist activity at mouse GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/chimeric Galphaq/i1 assessed as induction of ectodomain she...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Probable G-protein coupled receptor 34
(Homo sapiens (Human))
The University Of Tokyo
Curated by
ChEMBL
Ligand
BDBM50096349
(CHEBI:52649 | CHEMBL1742484)
Copy SMILES
Copy InChI
Affinity Data
EC50: 245nM
Assay Description:
Agonist activity at human GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/chimeric Galphaq/i1 assessed as induction of AP-TGFalpha re...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Putative P2Y purinoceptor 10
(Mus musculus)
The University Of Tokyo
Curated by
ChEMBL
Ligand
BDBM50096349
(CHEBI:52649 | CHEMBL1742484)
Copy SMILES
Copy InChI
Affinity Data
EC50: 20nM
Assay Description:
Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...
More data for this Ligand-Target Pair
Target Info
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Putative P2Y purinoceptor 10
(Mus musculus)
The University Of Tokyo
Curated by
ChEMBL
Ligand
BDBM50096349
(CHEBI:52649 | CHEMBL1742484)
Copy SMILES
Copy InChI
Affinity Data
EC50: 19nM
Assay Description:
Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...
More data for this Ligand-Target Pair
Target Info
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Probable G-protein coupled receptor 34
(Homo sapiens (Human))
The University Of Tokyo
Curated by
ChEMBL
Ligand
BDBM50096349
(CHEBI:52649 | CHEMBL1742484)
Copy SMILES
Copy InChI
Affinity Data
EC50: >3.00E+3nM
Assay Description:
Agonist activity at human GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Probable G-protein coupled receptor 34
(Homo sapiens (Human))
The University Of Tokyo
Curated by
ChEMBL
Ligand
BDBM50096349
(CHEBI:52649 | CHEMBL1742484)
Copy SMILES
Copy InChI
Affinity Data
EC50: >3.16E+3nM
Assay Description:
Agonist activity at human GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Probable G-protein coupled receptor 34
(Danio rerio)
The University Of Tokyo
Curated by
ChEMBL
Ligand
BDBM50096349
(CHEBI:52649 | CHEMBL1742484)
Copy SMILES
Copy InChI
Affinity Data
EC50: 130nM
Assay Description:
Agonist activity at zebrafish GPR34 type a expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain s...
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/TrEMBL
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Probable G-protein coupled receptor 34
(Danio rerio)
The University Of Tokyo
Curated by
ChEMBL
Ligand
BDBM50096349
(CHEBI:52649 | CHEMBL1742484)
Copy SMILES
Copy InChI
Affinity Data
EC50: 129nM
Assay Description:
Agonist activity at zebrafish GPR34 type a expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain s...
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/TrEMBL
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Probable G-protein coupled receptor 34
(Danio rerio)
The University Of Tokyo
Curated by
ChEMBL
Ligand
BDBM50096349
(CHEBI:52649 | CHEMBL1742484)
Copy SMILES
Copy InChI
Affinity Data
EC50: 3.5nM
Assay Description:
Agonist activity at zebrafish GPR34 type b expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain s...
More data for this Ligand-Target Pair
Target Info
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/TrEMBL
B.MOAD
DrugBank
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Probable G-protein coupled receptor 34
(Danio rerio)
The University Of Tokyo
Curated by
ChEMBL
Ligand
BDBM50096349
(CHEBI:52649 | CHEMBL1742484)
Copy SMILES
Copy InChI
Affinity Data
EC50: 3.5nM
Assay Description:
Agonist activity at zebrafish GPR34 type b expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain s...
More data for this Ligand-Target Pair
Target Info
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/TrEMBL
B.MOAD
DrugBank
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Probable G-protein coupled receptor 34
(Mus musculus)
The University Of Tokyo
Curated by
ChEMBL
Ligand
BDBM50096349
(CHEBI:52649 | CHEMBL1742484)
Copy SMILES
Copy InChI
Affinity Data
EC50: 230nM
Assay Description:
Agonist activity at mouse GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Probable G-protein coupled receptor 34
(Mus musculus)
The University Of Tokyo
Curated by
ChEMBL
Ligand
BDBM50096349
(CHEBI:52649 | CHEMBL1742484)
Copy SMILES
Copy InChI
Affinity Data
EC50: 234nM
Assay Description:
Agonist activity at mouse GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Probable G-protein coupled receptor 174
(Mus musculus)
The University Of Tokyo
Curated by
ChEMBL
Ligand
BDBM50096349
(CHEBI:52649 | CHEMBL1742484)
Copy SMILES
Copy InChI
Affinity Data
EC50: 34nM
Assay Description:
Agonist activity at mouse GPR174 transfected in human HEK293FT cells co-transfected with AP-TGFalpha assessed as AP-TGFalpha release incubated for 90...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
PubMed
Copy BDB DOI
Target
Putative P2Y purinoceptor 10
(Homo sapiens (Human))
The University Of Tokyo
Curated by
ChEMBL
Ligand
BDBM50096349
(CHEBI:52649 | CHEMBL1742484)
Copy SMILES
Copy InChI
Affinity Data
EC50: 28nM
Assay Description:
Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay
More data for this Ligand-Target Pair
Target Info
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI