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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 9 hits in this display   

TargetThymidine kinase 2, mitochondrial(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50100412(BDBM50206505 | CHEMBL392957 | Dodecanoic acid 4-hy...)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibitory concentration against mitochondrial thymidine kinase (TK-2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase 2, mitochondrial(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50100412(BDBM50206505 | CHEMBL392957 | Dodecanoic acid 4-hy...)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of human TK2 assessed as [methyl-3H]dThd phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxynucleoside kinase(Drosophila melanogaster)
Universit£

Curated by ChEMBL
LigandPNGBDBM50100412(BDBM50206505 | CHEMBL392957 | Dodecanoic acid 4-hy...)
Affinity DataIC50:  8.72E+5nMAssay Description:Inhibitory concentration against Drosophila melanogaster deoxyribonucleoside kinase (Dm-dNK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxynucleoside kinase(Drosophila melanogaster)
Universit£

Curated by ChEMBL
LigandPNGBDBM50100412(BDBM50206505 | CHEMBL392957 | Dodecanoic acid 4-hy...)
Affinity DataIC50:  8.72E+5nMAssay Description:Inhibition of Drosophila melanogaster dNK assessed as [methyl-3H]dThd phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase(Varicella-zoster virus (strain Dumas) (HHV-3) (Hum...)
Universit£

Curated by ChEMBL
LigandPNGBDBM50100412(BDBM50206505 | CHEMBL392957 | Dodecanoic acid 4-hy...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against Varicella- zoster virus thymidine kinase(VZV TK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50100412(BDBM50206505 | CHEMBL392957 | Dodecanoic acid 4-hy...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human TK1 assessed as [methyl-3H]dThd phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase(Varicella-zoster virus (strain Dumas) (HHV-3) (Hum...)
Universit£

Curated by ChEMBL
LigandPNGBDBM50100412(BDBM50206505 | CHEMBL392957 | Dodecanoic acid 4-hy...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of VZV TK assessed as [methyl-3H]dThd phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50100412(BDBM50206505 | CHEMBL392957 | Dodecanoic acid 4-hy...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against cytosolic thymidine kinase (TK-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Universit£

Curated by ChEMBL
LigandPNGBDBM50100412(BDBM50206505 | CHEMBL392957 | Dodecanoic acid 4-hy...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against Herpes simplex virus type 1 thymidine kinase(HSV-1 TK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed