Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetProbable G-protein coupled receptor 174(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL

LigandBDBM50096586(CHEMBL3577265)Copy SMILESCopy InChI

Affinity DataEC50:  31nMAssay Description:Agonist activity at GPR174 (unknown origin) transfected in HEK293FT cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLKEGGPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL

LigandBDBM50096586(CHEMBL3577265)Copy SMILESCopy InChI

Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair

Target InfoReactome pathway
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLKEGGPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetProbable G-protein coupled receptor 174(Mus musculus)
The University Of Tokyo

Curated by ChEMBL

LigandBDBM50096586(CHEMBL3577265)Copy SMILESCopy InChI

Affinity DataEC50:  34nMAssay Description:Agonist activity at mouse GPR174 transfected in human HEK293FT cells co-transfected with AP-TGFalpha assessed as AP-TGFalpha release incubated for 90...More data for this Ligand-Target Pair

Target InfoPDBMMDBKEGG
UniProtKB/SwissProt
B.MOADGoogleScholar

Ligand InfoCHEMBLKEGGPC cidPC sidSimilars

In DepthDetails PubMed
Copy BDB DOI

TargetProbable G-protein coupled receptor 174(Mus musculus)
The University Of Tokyo

Curated by ChEMBL

LigandBDBM50096586(CHEMBL3577265)Copy SMILESCopy InChI

Affinity DataEC50:  34nMAssay Description:Agonist activity at mouse GPR174 transfected in human HEK293FT cells co-transfected with AP-TGFalpha assessed as AP-TGFalpha release incubated for 90...More data for this Ligand-Target Pair

Target InfoPDBMMDBKEGG
UniProtKB/SwissProt
B.MOADGoogleScholar

Ligand InfoCHEMBLKEGGPC cidPC sidSimilars

In DepthDetails PubMed
Copy BDB DOI

TargetProbable G-protein coupled receptor 174(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL

LigandBDBM50096586(CHEMBL3577265)Copy SMILESCopy InChI

Affinity DataEC50:  31nMAssay Description:Agonist activity at GPR174 (unknown origin) transfected in HEK293FT cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLKEGGPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI