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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075897(CHEMBL84190 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-y...)
Affinity DataIC50:  380nMAssay Description:Binding affinity towards Beta-2 adrenergic receptor in CHO cells expressing the cloned human receptor using 1251-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075897(CHEMBL84190 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-y...)
Affinity DataIC50:  380nMAssay Description:Binding affinity towards human Beta-2 adrenergic receptor expressed in CHO cells, using [125I]-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075897(CHEMBL84190 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-y...)
Affinity DataIC50:  580nMAssay Description:Binding affinity towards Beta-1 adrenergic receptor in CHO cells expressing the cloned human receptor using 1251-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075897(CHEMBL84190 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-y...)
Affinity DataIC50:  580nMAssay Description:Binding affinity towards human Beta-1 adrenergic receptor expressed in CHO cells, using 1251-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075897(CHEMBL84190 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-y...)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity towards Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075897(CHEMBL84190 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-y...)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity towards Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075897(CHEMBL84190 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-y...)
Affinity DataEC50:  2.20nMAssay Description:In vitro effective concentration against beta-3 adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075897(CHEMBL84190 | N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-y...)
Affinity DataEC50:  4.57E+8nMAssay Description:In vitro effective concentration against beta-3 adrenergic receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed