Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50093040(CHEMBL74085 | N-[4-(6,7-Dihydroxy-1,2,3,4-tetrahyd...)
Affinity DataIC50:  200nMAssay Description:Compound was evaluated for its inhibitory activity against CHO cells expressing the cloned human Beta-1 adrenergic receptor in the presence of [125I]...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50093040(CHEMBL74085 | N-[4-(6,7-Dihydroxy-1,2,3,4-tetrahyd...)
Affinity DataIC50:  1.20E+3nMAssay Description:Compound was evaluated for its inhibitory activity against CHO cells expressing the cloned human Beta-1 adrenergic receptor in the presence of [125I]...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50093040(CHEMBL74085 | N-[4-(6,7-Dihydroxy-1,2,3,4-tetrahyd...)
Affinity DataEC50:  19nMAssay Description:Compound was evaluated for its inhibitory activity against human beta2 adrenergic receptor (AR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50093040(CHEMBL74085 | N-[4-(6,7-Dihydroxy-1,2,3,4-tetrahyd...)
Affinity DataEC50:  36nMAssay Description:Percent adenylyl cyclase activation at 10000 nM of compound concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50093040(CHEMBL74085 | N-[4-(6,7-Dihydroxy-1,2,3,4-tetrahyd...)
Affinity DataEC50:  66nMAssay Description:Inhibitory activity against human beta3 adrenergic receptor (AR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed