Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetChemerin-like receptor 1(Homo sapiens (Human))
Kyowa Kirin

Curated by ChEMBL
LigandPNGBDBM50517137(CHEMBL4457246)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of chemR23 in human CAL1 cells assessed as reduction in chemerin-induced intracellular calcium ion concentration preincubated for 45 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyowa Kirin

Curated by ChEMBL
LigandPNGBDBM50517137(CHEMBL4457246)
Affinity DataIC50:  9.90E+3nMAssay Description:Inhibition of CXCR4 expressed in human CAL1 cells assessed as reduction in SDF1alpha-induced intracellular calcium ion concentration preincubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChemerin-like receptor 1(Homo sapiens (Human))
Kyowa Kirin

Curated by ChEMBL
LigandPNGBDBM50517137(CHEMBL4457246)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at chemR23 expressed in human CAL1 cells assessed as increase in intracellular calcium ion concentrationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed