Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 79 hits in this display
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
IC50: 20nMAssay Description:Inhibition of human recombinant HDAC6 using ZMAL (Z-Lys(Ac)-AMC) fluorogenic substrate incubated for 90 mins by fluorescence based assayMore data for this Ligand-Target Pair
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
IC50: 25nMAssay Description:Inhibition of recombinant full length human N-terminal GST-tagged HDAC6 expressed in baculovirus infected sf9 insect cells pretreated with compound f...More data for this Ligand-Target Pair
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
IC50: 100nMAssay Description:Inhibition of tubastatin-Alexa647-tracer binding to recombinant GST-tagged HDAC10 (unknown origin) measured after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
IC50: 500nMAssay Description:Inhibition of human recombinant HDAC1 using ZMAL (Z-Lys(Ac)-AMC) fluorogenic substrate incubated for 90 mins by fluorescence based assayMore data for this Ligand-Target Pair
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
IC50: 3.02E+3nMAssay Description:HDAC inhibition assays were performed by Reaction Biology Corp. (Malvern, Pa.) using isolated human, recombinant full-length HDAC1 and -6 from a bacu...More data for this Ligand-Target Pair
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
IC50: 3.02E+3nMAssay Description:HDAC inhibition assays were performed by Reaction Biology Corp. (Malvern, Pa.) using isolated human, recombinant full-length HDAC1 and -6 from a bacu...More data for this Ligand-Target Pair
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
IC50: 3.02E+3nMAssay Description:Inhibition of human recombinant HDAC1 expressed in Sf9 cells incubated for 2 hrs using RHKK-Ac fluorogenic substrateMore data for this Ligand-Target Pair
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
IC50: 3.02E+3nMAssay Description:HDAC inhibition assays were performed by Reaction Biology Corp. (Malvern, Pa.) using isolated human, recombinant full-length HDAC1 and -6 from a bacu...More data for this Ligand-Target Pair
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
IC50: 3.02E+3nMpH: 8.0Assay Description:HDAC inhibition assays were performed by Reaction Biology Corp. (Malvern, Pa.) using isolated human, recombinant full-length HDAC1 and -6 from a bacu...More data for this Ligand-Target Pair
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
BDBM50398716(CHEMBL2179618 | US10227295, Compound 5g | US940985...)
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