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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
44
hits in this display
Target
5-hydroxytryptamine receptor 4
(GUINEA PIG)
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
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Affinity Data
Ki: 0.577nM
Assay Description:
Displacement of [3H]GR113808 from 5HT4 receptor in guinea pig striatal membranes
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 4
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 2nM
Assay Description:
Displacement of [3H]GR113808 from human recombinant 5HT4 receptor expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
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CHEMBL
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Target
D(4) dopamine receptor
(RAT)
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
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Affinity Data
Ki: 43nM
Assay Description:
Binding affinity to rat dopamine D4 receptor
More data for this Ligand-Target Pair
Target Info
Reactome pathway
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PC sid
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Target
Sigma non-opioid intracellular receptor 1
(RAT)
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
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Affinity Data
Ki: 60nM
Assay Description:
Binding affinity to rat sigma 1 receptor
More data for this Ligand-Target Pair
Target Info
PDB
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CHEMBL
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PC sid
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PubMed
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Target
5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 66nM
Assay Description:
Binding affinity to human 5-HT2B receptor
More data for this Ligand-Target Pair
Target Info
PDB
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KEGG
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CHEMBL
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PC sid
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Article
PubMed
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Target
D(2) dopamine receptor
(Rattus norvegicus (rat))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
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Affinity Data
Ki: 220nM
Assay Description:
Binding affinity to rat dopamine D2 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
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CHEMBL
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PC sid
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 300nM
Assay Description:
Binding affinity to human 5-HT1A receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
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Ligand Info
CHEMBL
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PC sid
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Article
PubMed
Copy BDB DOI
Target
D(3) dopamine receptor
(Rattus norvegicus (Rat))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
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Affinity Data
Ki: 336nM
Assay Description:
Binding affinity to rat dopamine D3 receptor
More data for this Ligand-Target Pair
Target Info
Reactome pathway
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CHEMBL
PC cid
PC sid
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Article
PubMed
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Target
Muscarinic acetylcholine receptor M2
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
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Affinity Data
Ki: 433nM
Assay Description:
Binding affinity to human muscarinic M2 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
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Target
5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 489nM
Assay Description:
Binding affinity to human 5-HT6 receptor
More data for this Ligand-Target Pair
Target Info
PDB
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KEGG
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CHEMBL
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Article
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Target
Alpha-1A adrenergic receptor
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
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Affinity Data
Ki: 522nM
Assay Description:
Binding affinity to human adrenergic alpha1A receptor
More data for this Ligand-Target Pair
Target Info
PDB
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KEGG
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CHEMBL
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Article
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Target
Alpha-2C adrenergic receptor
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 556nM
Assay Description:
Binding affinity to human adrenergic Alpha-2C receptor
More data for this Ligand-Target Pair
Target Info
PDB
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Target
Alpha-2B adrenergic receptor
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 671nM
Assay Description:
Binding affinity to human adrenergic alpha2B receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
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CHEMBL
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PC sid
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Article
PubMed
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Target
5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 685nM
Assay Description:
Binding affinity to human 5-HT2C receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
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GoogleScholar
Ligand Info
CHEMBL
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PC sid
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Details
Article
PubMed
Copy BDB DOI
Target
Muscarinic acetylcholine receptor M4
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 760nM
Assay Description:
Binding affinity to human muscarinic M4 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
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CHEMBL
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PC sid
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Article
PubMed
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Target
5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 820nM
Assay Description:
Binding affinity to human 5-HT1B receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Muscarinic acetylcholine receptor M3
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 823nM
Assay Description:
Binding affinity to human muscarinic M3 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
D(1B) dopamine receptor
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 972nM
Assay Description:
Binding affinity to human dopamine D5 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
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In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Muscarinic acetylcholine receptor M5
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 972nM
Assay Description:
Binding affinity to human muscarinic M5 receptor
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
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GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
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In Depth
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Article
PubMed
Copy BDB DOI
Target
5-hydroxytryptamine receptor 3A
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.07E+3nM
Assay Description:
Binding affinity to human 5-HT3 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
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In Depth
Details
Article
PubMed
Copy BDB DOI
Target
5-hydroxytryptamine receptor 1D
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.30E+3nM
Assay Description:
Binding affinity to human 5-HT1D receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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In Depth
Details
Article
PubMed
Copy BDB DOI
Target
5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.78E+3nM
Assay Description:
Binding affinity to human 5-HT2A receptor
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
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In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Sodium-dependent dopamine transporter
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 2.02E+3nM
Assay Description:
Binding affinity to human DAT
More data for this Ligand-Target Pair
Target Info
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
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In Depth
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Article
PubMed
Copy BDB DOI
Target
Alpha-2A adrenergic receptor
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 2.24E+3nM
Assay Description:
Binding affinity to human adrenergic alpha2A receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
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Ligand Info
CHEMBL
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PC sid
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In Depth
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Article
PubMed
Copy BDB DOI
Target
Alpha-1D adrenergic receptor
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 2.28E+3nM
Assay Description:
Binding affinity to human adrenergic Alpha-1D receptor
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
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GoogleScholar
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CHEMBL
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PC sid
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Article
PubMed
Copy BDB DOI
Target
D(1A) dopamine receptor
(RAT)
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 2.29E+3nM
Assay Description:
Binding affinity to rat dopamine D1 receptor
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Histamine H1 receptor
(Cavia porcellus (domestic guinea pig))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
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Affinity Data
Ki: 2.73E+3nM
Assay Description:
Binding affinity to guinea pig histamine H1 receptor
More data for this Ligand-Target Pair
Target Info
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Sodium-dependent noradrenaline transporter
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 3.23E+3nM
Assay Description:
Binding affinity to human NET
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
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In Depth
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Article
PubMed
Copy BDB DOI
Target
5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 5.70E+3nM
Assay Description:
Binding affinity to human 5-HT7 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
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antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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Article
PubMed
Copy BDB DOI
Target
5-hydroxytryptamine receptor 5A
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 8.59E+3nM
Assay Description:
Binding affinity to human 5-HT5A receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
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In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Sodium-dependent serotonin transporter
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 9.01E+3nM
Assay Description:
Binding affinity to human SERT
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
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GoogleScholar
Ligand Info
CHEMBL
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PC sid
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Details
Article
PubMed
Copy BDB DOI
Target
Alpha-1B adrenergic receptor
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
Assay Description:
Binding affinity to human adrenergic Alpha-1B receptor
More data for this Ligand-Target Pair
Target Info
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Delta-type opioid receptor
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Binding affinity to human delta opioid receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
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In Depth
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Article
PubMed
Copy BDB DOI
Target
5-hydroxytryptamine receptor 1E
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.00E+4nM
Assay Description:
Binding affinity to human 5-HT1E receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
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antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Muscarinic acetylcholine receptor M1
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
Assay Description:
Binding affinity to human muscarinic M1 receptor
More data for this Ligand-Target Pair
Target Info
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Mu-type opioid receptor
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
Assay Description:
Binding affinity to human mu opioid receptor
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
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In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Kappa-type opioid receptor
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
Assay Description:
Binding affinity to human kappa opioid receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
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In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Histamine receptor H4
(GUINEA PIG)
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Binding affinity to guinea pig histamine H4 receptor
More data for this Ligand-Target Pair
Target Info
UniProtKB/TrEMBL
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
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Article
PubMed
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Target
Histamine H3 receptor
(GUINEA PIG)
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Binding affinity to guinea pig histamine H3 receptor
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Histamine H2 receptor
(Cavia porcellus (domestic guinea pig))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
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Copy InChI
Affinity Data
Ki: >1.00E+4nM
Assay Description:
Binding affinity to guinea pig histamine H2 receptor
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Beta-1 adrenergic receptor
(Rattus norvegicus (Rat))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Binding affinity to rat adrenergic beta-1 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
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In Depth
Details
Article
PubMed
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Target
Beta-2 adrenergic receptor
(Rattus norvegicus)
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Binding affinity to rat adrenergic beta2 receptor
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Beta-3 adrenergic receptor
(Rattus norvegicus)
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
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Copy InChI
Affinity Data
Ki: >1.00E+4nM
Assay Description:
Binding affinity to rat adrenergic beta3 receptor
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
5-hydroxytryptamine receptor 4
(Homo sapiens (Human))
National Institute Of Mental Health
Curated by
ChEMBL
Ligand
BDBM50327860
((1-Butylpiperidin-4-yl)methyl 7-chloro-8-(methylam...)
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Affinity Data
EC50: 14nM
Assay Description:
Agonist activity at 5HT4 receptor expressed in HEK293/L9 cells by cAMP assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI