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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

TargetHistone deacetylase 3(Homo sapiens (Human))
Birla Institute Of Technology And Science-Pilani Hyderabad Campus

Curated by ChEMBL
LigandPNGBDBM50592234(CHEMBL5209383)
Affinity DataIC50:  15nMAssay Description:Inhibition of recombinant human HDAC3 using fluorescent as substrate measured for 15 mins by fluorescence based microtiter plate assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Birla Institute Of Technology And Science-Pilani Hyderabad Campus

Curated by ChEMBL
LigandPNGBDBM50592234(CHEMBL5209383)
Affinity DataIC50:  289nMAssay Description:Inhibition of recombinant human HDAC1 using fluorescent as substrate measured for 15 mins by fluorescence based microtiter plate assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Birla Institute Of Technology And Science-Pilani Hyderabad Campus

Curated by ChEMBL
LigandPNGBDBM50592234(CHEMBL5209383)
Affinity DataIC50:  534nMAssay Description:Inhibition of recombinant human HDAC2 using fluorescent as substrate measured for 30 mins by fluorescence based microtiter plate assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Birla Institute Of Technology And Science-Pilani Hyderabad Campus

Curated by ChEMBL
LigandPNGBDBM50592234(CHEMBL5209383)
Affinity DataIC50:  2.35E+3nMAssay Description:Inhibition of recombinant human HDAC8 using fluorescent as substrate measured for 10 mins by fluorescence based microtiter plate assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Birla Institute Of Technology And Science-Pilani Hyderabad Campus

Curated by ChEMBL
LigandPNGBDBM50592234(CHEMBL5209383)
Affinity DataIC50:  4.90E+4nMAssay Description:Inhibition of recombinant human HDAC6 using fluorescent as substrate measured for 10 mins by fluorescence based microtiter plate assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Birla Institute Of Technology And Science-Pilani Hyderabad Campus

Curated by ChEMBL
LigandPNGBDBM50592234(CHEMBL5209383)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant human HDAC4 using fluorescent as substrate measured for 30 mins by fluorescence based microtiter plate assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Birla Institute Of Technology And Science-Pilani Hyderabad Campus

Curated by ChEMBL
LigandPNGBDBM50592234(CHEMBL5209383)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant human HDAC5 using fluorescent as substrate measured for 30 mins by fluorescence based microtiter plate assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed