Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257302(2-(1-{3-[6-(Furan-3-carbonyl)-1-propyl-naphthalen-...)
Affinity DataEC50:  130nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257302(2-(1-{3-[6-(Furan-3-carbonyl)-1-propyl-naphthalen-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARdelta receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257302(2-(1-{3-[6-(Furan-3-carbonyl)-1-propyl-naphthalen-...)
Affinity DataEC50:  430nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed