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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
8
hits in this display
Target
AP2-associated protein kinase 1
(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by
ChEMBL
Ligand
BDBM50511383
(CHEMBL4531680)
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Affinity Data
Ki: 8.20nM
Assay Description:
Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...
More data for this Ligand-Target Pair
Target Info
PDB
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KEGG
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Target
BMP-2-inducible protein kinase
(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by
ChEMBL
Ligand
BDBM50511383
(CHEMBL4531680)
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Affinity Data
Ki: 20nM
Assay Description:
Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...
More data for this Ligand-Target Pair
Target Info
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KEGG
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antibodypedia
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Article
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Target
Serine/threonine-protein kinase 16
(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by
ChEMBL
Ligand
BDBM50511383
(CHEMBL4531680)
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Affinity Data
Ki: 310nM
Assay Description:
Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged STK16 kinase domain (13 to 305 residues) (unknown origin...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
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In Depth
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Target
Cyclin-G-associated kinase
(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by
ChEMBL
Ligand
BDBM50511383
(CHEMBL4531680)
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Affinity Data
Ki: 1.70E+3nM
Assay Description:
Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged GAK kinase domain (12 to 347 residues) (unknown origin) ...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
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KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
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PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
AP2-associated protein kinase 1
(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by
ChEMBL
Ligand
BDBM50511383
(CHEMBL4531680)
Copy SMILES
Copy InChI
Affinity Data
IC50: 375nM
Assay Description:
Inhibition of tracer K5 binding to N-terminal nano luciferase-fused AAK1 (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by N...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
BMP-2-inducible protein kinase
(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by
ChEMBL
Ligand
BDBM50511383
(CHEMBL4531680)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.89E+3nM
Assay Description:
Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Cyclin-G-associated kinase
(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by
ChEMBL
Ligand
BDBM50511383
(CHEMBL4531680)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of tracer K5 binding to N-terminal nano luciferase-fused GAK (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by Na...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Serine/threonine-protein kinase 16
(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by
ChEMBL
Ligand
BDBM50511383
(CHEMBL4531680)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of tracer K5 binding to N-terminal nano luciferase-fused STK16 (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI