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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 13 hits in this display   

Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50299166((6aR,9R)-N,N-diethyl-4,6,6a,7,8,9-hexahydroindolo[...)
Affinity DataIC50:  3nMAssay Description:Inhibition of 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50299166((6aR,9R)-N,N-diethyl-4,6,6a,7,8,9-hexahydroindolo[...)
Affinity DataIC50:  6nMAssay Description:Inhibition of 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50299166((6aR,9R)-N,N-diethyl-4,6,6a,7,8,9-hexahydroindolo[...)
Affinity DataIC50:  16nMAssay Description:Inhibition of 5HT6 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50299166((6aR,9R)-N,N-diethyl-4,6,6a,7,8,9-hexahydroindolo[...)
Affinity DataIC50:  54nMAssay Description:Inhibition of 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50299166((6aR,9R)-N,N-diethyl-4,6,6a,7,8,9-hexahydroindolo[...)
Affinity DataIC50:  143nMAssay Description:Inhibition of 5HT7 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50299166((6aR,9R)-N,N-diethyl-4,6,6a,7,8,9-hexahydroindolo[...)
Affinity DataIC50:  1.29E+3nMAssay Description:Inhibition of 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50299166((6aR,9R)-N,N-diethyl-4,6,6a,7,8,9-hexahydroindolo[...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of adrenergic beta1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50299166((6aR,9R)-N,N-diethyl-4,6,6a,7,8,9-hexahydroindolo[...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of dopamine D3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50299166((6aR,9R)-N,N-diethyl-4,6,6a,7,8,9-hexahydroindolo[...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50299166((6aR,9R)-N,N-diethyl-4,6,6a,7,8,9-hexahydroindolo[...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of adrenergic alpha2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50299166((6aR,9R)-N,N-diethyl-4,6,6a,7,8,9-hexahydroindolo[...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of adrenergic alpha2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50299166((6aR,9R)-N,N-diethyl-4,6,6a,7,8,9-hexahydroindolo[...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]I-TAC from human CXCR3 expressed in CHO cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50299166((6aR,9R)-N,N-diethyl-4,6,6a,7,8,9-hexahydroindolo[...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed