Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Sanofi Research

Curated by ChEMBL

LigandBDBM50395750(CHEMBL2164508)Copy SMILESCopy InChI

Affinity DataKi:  286nMAssay Description:Displacement of [125I]-ghrelin from human GHSR1 expressed in CHO-CREluc cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Sanofi Research

Curated by ChEMBL

LigandBDBM50395750(CHEMBL2164508)Copy SMILESCopy InChI

Affinity DataIC50:  129nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI