Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 12 hits in this display   

Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

Curated by ChEMBL
LigandPNGBDBM50148832(CHEMBL3771331)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) after 1.5 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

Curated by ChEMBL
LigandPNGBDBM50148832(CHEMBL3771331)
Affinity DataKi:  427nMAssay Description:Displacement of [3H]LSD from 5-HT7A receptor (unknown origin) after 1.5 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

Curated by ChEMBL
LigandPNGBDBM50148832(CHEMBL3771331)
Affinity DataKi:  994nMAssay Description:Displacement of [3H]LSD from 5-HT5A receptor (unknown origin) after 1.5 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

Curated by ChEMBL
LigandPNGBDBM50148832(CHEMBL3771331)
Affinity DataKi:  1.31E+3nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2A receptor (unknown origin) after 1.5 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

Curated by ChEMBL
LigandPNGBDBM50148832(CHEMBL3771331)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [3H]LSD from 5-HT2C receptor (unknown origin) after 1.5 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

Curated by ChEMBL
LigandPNGBDBM50148832(CHEMBL3771331)
Affinity DataKi:  5.91E+3nMAssay Description:Displacement of [3H]LSD from 5-HT6 receptor (unknown origin) after 1.5 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

Curated by ChEMBL
LigandPNGBDBM50148832(CHEMBL3771331)
Affinity DataKi:  6.76E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor (unknown origin) after 1.5 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

Curated by ChEMBL
LigandPNGBDBM50148832(CHEMBL3771331)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-5-HT from 5-HT1E receptor (unknown origin) after 1.5 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

Curated by ChEMBL
LigandPNGBDBM50148832(CHEMBL3771331)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]GR127543 from 5-HT1D receptor (unknown origin) after 1.5 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

Curated by ChEMBL
LigandPNGBDBM50148832(CHEMBL3771331)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]LY278584 from 5-HT3 receptor (unknown origin) after 1.5 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

Curated by ChEMBL
LigandPNGBDBM50148832(CHEMBL3771331)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]GR127543 from 5-HT1B receptor (unknown origin) after 1.5 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

Curated by ChEMBL
LigandPNGBDBM50148832(CHEMBL3771331)
Affinity DataIC50:  104nMAssay Description:Antagonist activity at 5-HT2B receptor (unknown origin) expressed in CHO-K1 cells assessed as calcium flux after 60 mins by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed