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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50244589(1-[6-(4-Methanesulfonyl-phenylamino)-5-nitro-pyrim...)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at GPR119 (unknown origin) expressed in HEK293 cells assessed as cAMP level by flash plate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed