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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetCathepsin S(Homo sapiens (Human))
National Tsing Hua University

Curated by ChEMBL
LigandPNGBDBM50320035(CHEMBL1083318 | Glycine, N-[(3S)-4-Benzyloxy-3-[[[...)
Affinity DataIC50:  4.40nMAssay Description:Inhibition of human recombinant cathepsin S expressed in Escherichia coli BL21 (DE3) after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
National Tsing Hua University

Curated by ChEMBL
LigandPNGBDBM248155(Cathepsin S inhibitor alpha-ketoamide, 6a)
Affinity DataIC50:  4.40nMpH: 6.5 T: 2°CAssay Description:A microplate-based screening procedure was used to study the effect of inhibition of re-Cat S, re-Cat L and re-Cat K on several compounds. The assays...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed